SCHEMBL24089986

SCHEMBL24089986

O=c1c2ccccc2nc(Nc2ccc(CO)cc2)n1-c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 1/20 0.55
PDE7A Q13946 2/20 0.51
RAB9A P51151 2/20 0.50
MDM2 Q00987 1/20 0.50
MAPT P10636 5/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
USP2 O75604 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24090010 0.91 USP2 (0.52) PDE7ARAB9AMAPTUSP2NPC1
SCHEMBL24089988 0.87 PIK3CD (0.46) ALOX12PDE7ARAB9AMDM2
SCHEMBL24090014 0.87 MAT2A (0.44) ALOX12
SCHEMBL24089947 0.87 ALOX12 (0.55) ALOX12PDE7ARAB9AMDM2MAPT
SCHEMBL24090113 0.85 ALOX12 (0.50) ALOX12PDE7ARAB9AMDM2MAPT
SCHEMBL24110995 0.84 ALOX12 (0.57) ALOX12PDE7ARAB9AMDM2MAPT
SCHEMBL24090115 0.81 ALDH1A1 (0.48) PDE7ARAB9AMAPTSMN1; SMN2USP2
SCHEMBL24090012 0.79 TOP2A (0.60) PDE7ARAB9AMAPTUSP2NPC1
SCHEMBL23045330 0.78 KDM4E (0.44)
SCHEMBL29623225 0.78 KDM4E (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11352366-B2 2-aminoquinazolinone derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-06-07 US disclosed
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-05-12 US disclosed
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, CRKL ALOX12 3008/4885PDE7A 2489/4885RAB9A 1045/4885
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, SLC26A3 ALOX12 3295/4885PDE7A 2591/4885RAB9A 902/4885
US-11352366-B2 2-aminoquinazolinone derivative CNKSR1, HAX1, SLC26A3 ALOX12 3295/4885PDE7A 2591/4885RAB9A 902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.