SCHEMBL2409149

SCHEMBL2409149

CN(Cc1cn(S(=O)(=O)c2cnn(C(F)F)c2)c(-c2cccnc2F)c1F)C(=O)OC(C)(C)C

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.32
KAT6A Q92794 1/20 0.31
KAT5 Q92993 1/20 0.31
RORC P51449 1/20 0.30
HTR2C P28335 2/20 0.30
SLC6A4 P31645 2/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30
MMP13 P45452 1/20 0.30
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2413759 0.90 RORC (0.36) KAT6AKAT5RORCHTR2CSLC6A4
SCHEMBL2417223 0.89 JAK3 (0.35) KAT6AKAT5RORCHTR2CSLC6A4
SCHEMBL5003076 0.88 BRD4 (0.34) BRD4MMP2MMP9MMP8MMP13
SCHEMBL2411042 0.87 HTR6 (0.33) KAT6AKAT5RORCHTR2CSLC6A4
SCHEMBL1833792 0.86 KAT6A (0.32) KAT6AKAT5HTR2CSLC6A4MMP2
SCHEMBL2409441 0.86 HTR2C (0.35) KAT6AKAT5HTR2CSLC6A4MMP2
SCHEMBL1832149 0.85 HTR2C (0.33) KAT6AKAT5RORCHTR2CSLC6A4
SCHEMBL4420269 0.85 HTR6 (0.37) HTR2CSLC6A4HTR2A
SCHEMBL1834426 0.84 HTR2C (0.33) KAT6AKAT5HTR2CSLC6A4HTR2A
SCHEMBL4570001 0.84 OXTR (0.34) KAT6AKAT5RORCHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed