SCHEMBL2410593

SCHEMBL2410593

CC(C)(C)C(Cc1cn(S(=O)(=O)N2CCOCC2)c(-c2cccnc2F)c1F)NC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.34
LIPG Q9Y5X9 1/20 0.34
HTT P42858 2/20 0.33
MEN1 O00255 2/20 0.33
ATM Q13315 1/20 0.33
ALDH1A1 P00352 5/20 0.33
CNR1 P21554 4/20 0.33
CNR2 P34972 3/20 0.33
MAPT P10636 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
OPRK1 P41145 1/20 0.32
USP2 O75604 1/20 0.32
NPC1 O15118 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2407099 0.93 OPRM1 (0.32) ALDH1A1KDM4ELMNAOPRK1SMN1; SMN2
SCHEMBL2409041 0.92 OPRM1 (0.32) KMT2AHTTMEN1ALDH1A1CNR2
Hydrochloric Acid SCHEMBL4420968 0.89 OPRM1 (0.31) OPRK1
Hydrochloric Acid SCHEMBL4422137 0.88 OPRM1 (0.31) OPRK1
SCHEMBL2410800 0.83
SCHEMBL2192366 0.83 DCTPP1 (0.31)
SCHEMBL2409724 0.82 PTGS2 (0.34) KMT2AMEN1
SCHEMBL2410511 0.82 ABCC9 (0.33) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL2194609 0.82 MMP2 (0.30)
SCHEMBL2411544 0.82 MMP2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed