SCHEMBL24106959

SCHEMBL24106959

NC(=S)N1CCC2(CC1)NCC(=O)N2Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.39
CYP2D6 P10635 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 2/20 0.38
CYP3A4 P08684 2/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
USP2 O75604 1/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM3 P20309 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24106950 0.89 OPRD1 (0.46) RIPK1CYP2D6ALDH1A1MAPK1CYP3A4
SCHEMBL15423927 0.83 ALDH1A1 (0.47) ALDH1A1KDM4ELMNAHTTMEN1
Simufilam SCHEMBL12627054 0.81 MC4R (0.46) ALDH1A1MAPK1GSK3AGSK3BKDM4E
SCHEMBL12656278 0.80 GSK3A (0.42) ALDH1A1GSK3AGSK3BKDM4ELMNA
Simufilam SCHEMBL22361808 0.80 MC4R (0.45) ALDH1A1MAPK1GSK3AGSK3BKDM4E
Simufilam SCHEMBL22361802 0.80 MC4R (0.45) ALDH1A1MAPK1GSK3AGSK3BKDM4E
SCHEMBL15423926 0.80 FAAH (0.56) CYP2D6ALDH1A1CYP3A4KDM4EOPRD1
Simufilam SCHEMBL22361805 0.79 MC4R (0.44) ALDH1A1MAPK1GSK3AGSK3BKDM4E
SCHEMBL15426043 0.79 ALDH1A1 (0.43) CYP2D6ALDH1A1CYP3A4KDM4ELMNA
SCHEMBL15423954 0.79 DRD4 (0.46) CYP2D6ALDH1A1GSK3AGSK3BUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210389298-A1 Alzheimer's Disease Assay in a Living Patient PAIN THERAPEUTICS, INC. (US) 2021-12-16 US disclosed