SCHEMBL24106950

SCHEMBL24106950

NC(=O)N1CCC2(CC1)NCC(=O)N2Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 1/20 0.44
RIPK1 Q13546 1/20 0.43
AMPD2 Q01433 2/20 0.41
CYP2D6 P10635 7/20 0.41
CYP3A4 P08684 3/20 0.41
USP2 O75604 1/20 0.41
MAPK1 P28482 1/20 0.41
CHRM2 P08172 3/20 0.40
CHRM3 P20309 1/20 0.40
LTA4H P09960 1/20 0.39
TSHR P16473 2/20 0.39
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24106959 0.89 RIPK1 (0.39) OPRD1OPRK1ALDH1A1KDM4ERIPK1
SCHEMBL15423926 0.83 FAAH (0.56) OPRD1OPRK1ALDH1A1KDM4ECYP2D6
Simufilam SCHEMBL12627054 0.82 MC4R (0.46) ALDH1A1KDM4EGAAMAPK1GSK3A
SCHEMBL1801385 0.82 RIPK1 (0.52) ALDH1A1KDM4ERIPK1CYP2D6CYP3A4
SCHEMBL4001000 0.82 L3MBTL1 (0.43) OPRD1OPRK1ALDH1A1KDM4EGAA
SCHEMBL12656278 0.81 GSK3A (0.42) OPRD1OPRK1ALDH1A1KDM4EGAA
Simufilam SCHEMBL22361808 0.81 MC4R (0.45) ALDH1A1KDM4EGAAMAPK1GSK3A
Simufilam SCHEMBL22361802 0.81 MC4R (0.45) ALDH1A1KDM4EGAAMAPK1GSK3A
SCHEMBL12627087 0.81 OPRD1 (0.51) OPRD1OPRK1ALDH1A1GAACYP2D6
SCHEMBL5152604 0.80 HDAC1 (0.45) OPRD1ALDH1A1KDM4EGAAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210389298-A1 Alzheimer's Disease Assay in a Living Patient PAIN THERAPEUTICS, INC. (US) 2021-12-16 US disclosed