SCHEMBL24166156

SCHEMBL24166156

COCCn1cnc2ccc(N)c(-c3ccc(OC)nc3)c2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.43
MTOR P42345 2/20 0.43
GRM2 Q14416 1/20 0.40
SYK P43405 3/20 0.39
P2RX3 P56373 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
ALOX15 P16050 1/20 0.37
BRAF P15056 1/20 0.36
PIK3CD O00329 2/20 0.35
PIK3CB P42338 2/20 0.35
PI4KA P42356 2/20 0.35
PIK3CG P48736 2/20 0.35
PI4KB Q9UBF8 2/20 0.35
PIP5K1C O60331 1/20 0.35
MAPK1 P28482 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30656840 1.00 PIK3CA (0.43) PIK3CAMTORGRM2SYKP2RX3
SCHEMBL24166480 0.86 ALOX15 (0.46) P2RX3KMT2AMEN1TDP1ALOX15
SCHEMBL30656834 0.86 ALOX15 (0.46) P2RX3KMT2AMEN1TDP1ALOX15
SCHEMBL30656795 0.84 BRAF (0.41) PIK3CASYKKMT2AMEN1BRAF
SCHEMBL24165960 0.84 BRAF (0.41) PIK3CASYKKMT2AMEN1BRAF
SCHEMBL24166503 0.84 ALDH1A1 (0.43) KMT2AMEN1TDP1BRAFMAPK1
SCHEMBL30656811 0.84 ALDH1A1 (0.43) KMT2AMEN1TDP1BRAFMAPK1
SCHEMBL24166121 0.83 CLK1 (0.43) GRM2P2RX3KMT2AMEN1TDP1
SCHEMBL30656848 0.83 CLK1 (0.43) GRM2P2RX3KMT2AMEN1TDP1
SCHEMBL24166155 0.83 KMT2A (0.40) SYKP2RX3KMT2AMEN1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357165-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2023-11-09 US disclosed
US-20230357165-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2023-11-09 US disclosed
US-20230357165-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2023-11-09 US disclosed
WO-2022003712-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2022-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230357165-A1 QUINAZOLINONES DERIVATIVES FOR TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE, PREPARATION AND USE THEREOF ATG7, GOT1, LIPC PIK3CA 2562/4885MTOR 730/4885GRM2 4328/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.