SCHEMBL24201256

SCHEMBL24201256

O=C(O)COCCNC(=O)CC12CC3CC4CC(C1)C2(C4)C3

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 8/20 0.41
ALDH1A1 P00352 4/20 0.38
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
OPRK1 P41145 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.32
PTP4A3 O75365 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24201351 0.98 EPHX2 (0.43) EPHX2ALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL24201251 0.98 EPHX2 (0.43) EPHX2ALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL24201339 0.86 EPHX2 (0.45) EPHX2ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL24201248 0.86 EPHX2 (0.45) EPHX2ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL24201335 0.81 ALDH1A1 (0.59) EPHX2ALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL24201206 0.81 ALDH1A1 (0.45) EPHX2ALDH1A1CYP3A4CYP2C19MEN1
SCHEMBL17457697 0.79 ALDH1A1 (0.60) EPHX2ALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL24201255 0.77 EPHX2 (0.60) EPHX2ALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL24201216 0.74 OPRK1 (0.32) OPRK1
SCHEMBL7778418 0.71 KDM4E (0.64) EPHX2ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3618833-B1 TRIPARTITE ANDROGEN RECEPTOR ELIMINATORS, METHODS AND USES THEREOF SPG THERAPEUTICS INC (US) 2022-01-19 EP disclosed