SCHEMBL24251660

SCHEMBL24251660

Nc1ccc(Br)nc1OCC(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
THRB P10828 1/20 0.42
G6PD P11413 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ADORA2A P29274 1/20 0.42
MBOAT4 Q96T53 3/20 0.36
SCN9A Q15858 2/20 0.34
HRH4 Q9H3N8 1/20 0.33
AMD1 P17707 1/20 0.33
NUDT1 P36639 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29392742 1.00 L3MBTL1 (0.42) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL21756757 0.79 ALDH1A1 (0.42) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL17490419 0.79 MAPT (0.42) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL3134237 0.77 ADORA2A (0.46) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL7016888 0.77 HPGD (0.42) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL22475331 0.74 ALDH1A1 (0.38) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL21756758 0.74 ALDH1A1 (0.41) L3MBTL1ALDH1A1MAPTMEN1KMT2A
SCHEMBL29391783 0.73 TXNRD1 (0.38) ALDH1A1ADORA2ACNR2
SCHEMBL24251675 0.73 TXNRD1 (0.38) ALDH1A1ADORA2ACNR2
SCHEMBL21223041 0.72 MBOAT4 (0.46) L3MBTL1ALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115701429-B 4- (1H-indol-1-yl) pyrimidine-2-amino derivative, and preparation method and application thereof 上海和誉生物医药科技有限公司 2024-03-12 CN disclosed
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
CN-115701429-A 4- (1H-indole-1-yl) pyrimidine-2-amino derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-02-10 CN disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed