SCHEMBL24251711

SCHEMBL24251711

CC(=O)Nc1cc([N+](=O)[O-])c(N2CCCC2)nc1OCC(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPK1 P28482 3/20 0.41
HTT P42858 1/20 0.41
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
GALR2 O43603 1/20 0.41
MITF O75030 1/20 0.41
LMNA P02545 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HPGD P15428 1/20 0.41
XBP1 P17861 1/20 0.41
CCR6 P51684 1/20 0.41
MAPT P10636 6/20 0.38
TDP1 Q9NUW8 3/20 0.38
CNR2 P34972 1/20 0.37
AR P10275 2/20 0.37
OPRK1 P41145 1/20 0.36
KMT2A Q03164 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28510516 0.91 ALDH1A1 (0.44) ALDH1A1MAPK1POLBSMN1; SMN2NPSR1
SCHEMBL29133283 0.85 WDR5 (0.40) ALDH1A1MAPK1POLBSMN1; SMN2NPSR1
SCHEMBL28973029 0.85 MCHR1 (0.38) ALDH1A1MAPK1POLBSMN1; SMN2NPSR1
SCHEMBL24251673 0.84 ALDH1A1 (0.44) ALDH1A1MAPK1HTTPOLBSMN1; SMN2
SCHEMBL17490379 0.83 NPSR1 (0.46) ALDH1A1HTTPOLBSMN1; SMN2NPSR1
SCHEMBL29389430 0.81 NPSR1 (0.46) ALDH1A1HTTPOLBSMN1; SMN2NPSR1
SCHEMBL24251729 0.81 NPSR1 (0.46) ALDH1A1HTTPOLBSMN1; SMN2NPSR1
SCHEMBL24251659 0.80 ALDH1A1 (0.44) ALDH1A1MAPK1HTTPOLBSMN1; SMN2
SCHEMBL18978915 0.75 ALDH1A1 (0.40) ALDH1A1POLBSMN1; SMN2NPSR1GALR2
SCHEMBL28973006 0.75 ALDH1A1 (0.45) ALDH1A1MAPK1HTTPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed