SCHEMBL24252550

SCHEMBL24252550

Cc1cccc(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.40
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
CYP2A6 P11509 1/20 0.39
CYP2B6 P20813 1/20 0.39
ENPP1 P22413 3/20 0.39
KIF11 P52732 1/20 0.39
PDK2 Q15119 1/20 0.39
AR P10275 1/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ESR2 Q92731 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29391919 1.00 HSD11B1 (0.40) HSD11B1PDCD1CD274CYP2A6CYP2B6
SCHEMBL27747416 0.83 PDCD1 (0.41) HSD11B1PDCD1CD274CYP2A6CYP2B6
SCHEMBL4090283 0.78 CYP2A6 (0.43) HSD11B1CYP2A6PDK2TSHRALDH1A1
SCHEMBL21357712 0.78 TRPA1 (0.49) CYP2A6ENPP1KIF11PDK2TSHR
SCHEMBL2597833 0.78 HSD11B1 (0.51) HSD11B1ENPP1KIF11PDK2AR
SCHEMBL28160333 0.77 PTGS2 (0.47) HPGDRAB9AHSD17B10TACR1
SCHEMBL5132773 0.76 ALDH1A1 (0.56) ENPP1KIF11PDK2ARTSHR
SCHEMBL27926229 0.76 ALDH1A1 (0.56) HSD11B1CYP2A6ENPP1KIF11PDK2
SCHEMBL27907878 0.76 CYP2A6 (0.56) HSD11B1CYP2A6ENPP1KIF11PDK2
SCHEMBL3793637 0.76 ALDH1A1 (0.56) CYP2A6ENPP1KIF11PDK2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303494-A1 BENZYLAMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF ACADEMY OF MILITARY MEDICAL SCIENCES (CN) 2023-09-28 US disclosed
US-20230303494-A1 BENZYLAMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF ACADEMY OF MILITARY MEDICAL SCIENCES (CN) 2023-09-28 US disclosed
EP-4198017-A1 BENZYLAMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF Academy of Military Medical Sciences (CN) 2023-06-21 EP disclosed
WO-2022033303-A1 BENZYLAMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 中国人民解放军军事科学院军事医学研究院 2022-02-17 WO disclosed
CN-109305934-A Phenylate analog derivative and officinal salt, purposes pharmaceutically 成都海博锐药业有限公司 2019-02-05 CN disclosed
CN-105143193-B Biaryl or heterocyclic biaryl substituted cyclohexene derivative compounds as CETP inhibitors 株式会社钟根堂 2017-12-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303494-A1 BENZYLAMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF CD274, PDCD1, PDCD1LG2 HSD11B1 452/4885PDCD1 2/4885CD274 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.