SCHEMBL2425876

SCHEMBL2425876

N#Cc1cncc(Oc2ccc(F)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
CYP19A1 P11511 1/20 0.49
SLC22A12 Q96S37 1/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 1/20 0.44
SLC6A3 Q01959 1/20 0.44
GRM5 P41594 2/20 0.43
NPY5R Q15761 1/20 0.43
XDH P47989 1/20 0.43
CYP2C19 P33261 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
VEGFA P15692 2/20 0.40
EPAS1 Q99814 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2422932 0.87 CHRNB2 (0.48) CYP3A4CYP19A1SLC22A12CHRNB2CHRNA4
SCHEMBL30689372 0.83 CYP19A1 (0.57) CYP3A4CYP19A1SLC22A12GRM5CYP11B1
SCHEMBL27368527 0.83 CYP19A1 (0.57) CYP3A4CYP19A1SLC22A12GRM5CYP11B1
SCHEMBL6821689 0.83 CYP19A1 (0.56) CYP3A4CYP19A1SLC22A12CHRNB2CHRNA4
SCHEMBL876009 0.80 CYP19A1 (0.45) CYP3A4CYP19A1GRM5VEGFAEPAS1
SCHEMBL876496 0.80 LTA4H (0.46) CYP3A4CYP19A1GRM5CYP11B1CYP11B2
SCHEMBL3138833 0.78 PARP15 (0.53) CYP3A4CYP19A1CYP1A2CYP2C19KDM4E
SCHEMBL16834849 0.77 SLC22A12 (0.43) CYP3A4SLC22A12CHRNB2CHRNA4NPY5R
SCHEMBL2196501 0.77 CYP19A1 (0.71) CYP19A1GRM5CYP11B1CYP11B2ALDH1A1
SCHEMBL923535 0.76 ALOX5 (0.50) CYP3A4CYP19A1SLC22A12CYP1A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011117254-A1 PIPERIDINE AMIDES AS MODULATORS OF THE GHRELIN RECEPTOR PROSIDION LIMITED (GB) 2011-09-29 WO disclosed