SCHEMBL24313221

SCHEMBL24313221

Cc1cc(N2CCCCCC2c2ccncc2)ncn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.43
CYP17A1 P05093 1/20 0.41
HDAC8 Q9BY41 1/20 0.39
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
PRCP P42785 1/20 0.36
CFB P00751 1/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24654724 0.88 PSEN1 (0.39) CYP17A1JAK2JAK3PSEN1PSEN2
SCHEMBL29456545 0.80 CRHBP (0.51) HDAC6HDAC8PRMT5WDR77CFB
SCHEMBL21516990 0.80 CRHBP (0.51) HDAC6HDAC8PRMT5WDR77CFB
SCHEMBL24313136 0.77 PRCP (0.41) CYP17A1PRCPMAPTL3MBTL1KDM4E
SCHEMBL24313222 0.76 JAK2 (0.35) CYP17A1JAK2JAK3PRCPMAPT
SCHEMBL30745929 0.74 HDAC6 (0.49) HDAC6HDAC8MAPTL3MBTL1KDM4E
SCHEMBL24313474 0.73 PRCP (0.43) CYP17A1PRCPMAPTLMNASMN1; SMN2
SCHEMBL20575880 0.71 PRCP (0.42) JAK2JAK3PSEN1PSEN2APH1B
SCHEMBL12090442 0.70 CHRNB2 (0.64) MAPTKDM4ELMNACHRNB2CHRNA7
SCHEMBL21516330 0.68 CRHBP (0.52) MAPTL3MBTL1KDM4EHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3784666-B1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2022-03-16 EP disclosed