SCHEMBL24313222

SCHEMBL24313222

CCc1ncccc1C1CCCCCN1c1cc(C)ncn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 4/20 0.35
JAK3 P52333 1/20 0.35
CYP17A1 P05093 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NTRK1 P04629 4/20 0.33
PRCP P42785 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HCRTR1 O43613 2/20 0.32
HCRTR2 O43614 2/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32
CXCR4 P61073 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24313136 0.80 PRCP (0.41) CYP17A1KDM4EMAPTL3MBTL1PRCP
SCHEMBL24313221 0.76 HDAC6 (0.43) JAK2JAK3CYP17A1KDM4EMAPT
SCHEMBL29456608 0.75 CRHBP (0.43) JAK2KDM4EMAPTL3MBTL1NTRK1
SCHEMBL31472394 0.75 CRHBP (0.43) JAK2KDM4EMAPTL3MBTL1NTRK1
SCHEMBL21516598 0.75 CRHBP (0.43) JAK2KDM4EMAPTL3MBTL1NTRK1
SCHEMBL24654724 0.74 PSEN1 (0.39) JAK2JAK3CYP17A1KDM4EMAPT
SCHEMBL24313474 0.72 PRCP (0.43) CYP17A1MAPTPRCPMEN1KMT2A
SCHEMBL9385174 0.71 CHRNB2 (0.49) MAPTLMNA
SCHEMBL11273849 0.71 CHRNB2 (0.49) MAPTLMNA
SCHEMBL21516627 0.70 CRHBP (0.47) JAK2KDM4EMAPTL3MBTL1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4043460-A1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF Merck Patent GmbH (DE) 2022-08-17 EP disclosed
EP-3784666-B1 ANTIPROLIFERATION COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2022-03-16 EP disclosed