SCHEMBL24316427

SCHEMBL24316427

COc1cc(Oc2ccc3ncc(C)c(=O)n3c2)cnc1OCc1ccc(C2CC2(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 5/20 0.42
PIK3CA P42336 3/20 0.35
MTOR P42345 3/20 0.35
RXFP1 Q9HBX9 1/20 0.33
KIT P10721 1/20 0.31
PDE1A P54750 5/20 0.31
PDE1B Q01064 5/20 0.31
PDE1C Q14123 5/20 0.31
ALKBH1 Q13686 2/20 0.31
KCNA5 P22460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24316587 0.88 CSF1R (0.44) CSF1RPIK3CAMTORRXFP1
SCHEMBL24316446 0.88 CSF1R (0.42) CSF1RPIK3CAMTORRXFP1PDE1A
SCHEMBL24316434 0.87 CSF1R (0.53) CSF1RPIK3CAMTORRXFP1KIT
SCHEMBL24316982 0.86 CSF1R (0.48) CSF1RPIK3CAMTORRXFP1KIT
SCHEMBL24316814 0.85 CSF1R (0.47) CSF1RPIK3CAMTORRXFP1
SCHEMBL24316983 0.84 CSF1R (0.46) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316448 0.83 CSF1R (0.45) CSF1RPIK3CAMTORRXFP1PDE1A
SCHEMBL24316437 0.82 CSF1R (0.45) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316429 0.82 CSF1R (0.40) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316553 0.82 CSF1R (0.46) CSF1RPIK3CAMTORRXFP1PDE1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057895-A1 HETEROAROMATIC COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2022-03-24 WO disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed