SCHEMBL24323964

SCHEMBL24323964

COC(=O)/C(=C\CC(C)(C)F)NC(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.33
CA12 O43570 2/20 0.33
CA14 Q9ULX7 2/20 0.33
APLNR P35414 1/20 0.33
CTSK P43235 9/20 0.33
TDP1 Q9NUW8 1/20 0.33
CA1 P00915 2/20 0.32
CA7 P43166 2/20 0.32
DGAT1 O75907 1/20 0.32
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
CTSS P25774 1/20 0.31
BTN3A1 O00481 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29601090 1.00 CA2 (0.33) CA2CA12CA14APLNRCTSK
SCHEMBL26838901 0.87 CA12 (0.35) CA2CA12CA14APLNRCTSK
SCHEMBL24298555 0.87 CA12 (0.35) CA2CA12CA14APLNRCTSK
SCHEMBL3863085 0.83 CA12 (0.35) CA2CA12CA14APLNRCTSK
SCHEMBL19519894 0.81 CTSK (0.33) CA2CA12CA14APLNRCTSK
SCHEMBL5787436 0.79 DGAT1 (0.38) CA2CA12CA14CTSKTDP1
SCHEMBL5787433 0.79 DGAT1 (0.38) CA2CA12CA14CTSKTDP1
SCHEMBL28673190 0.79 CA12 (0.31) CA2CA12CA14
SCHEMBL12903905 0.78 CA2 (0.32) CA2CA12CA14CTSKTDP1
SCHEMBL19519893 0.78 ALDH1A1 (0.33) CA2CA12CA14CTSKTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023196429-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-12 WO disclosed
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed