SCHEMBL24324093

SCHEMBL24324093

OCc1cncc(N2CCCCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.46
TRPV3 Q8NET8 2/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
SORD Q00796 2/20 0.38
PIM2 Q9P1W9 2/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP1A2 P05177 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTR1A P08908 1/20 0.38
HPGD P15428 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PIM1 P11309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24922389 0.83 ALDH1A1 (0.40) CYP11B1CYP11B2PIM2KMT2AMEN1
SCHEMBL2724262 0.83 HTR2C (0.58) PIM2KMT2AMEN1CYP3A4CYP2C9
SCHEMBL16366822 0.81 PDE10A (0.51) PDE10ATRPV3CYP11B1CYP11B2PIM2
SCHEMBL15537495 0.75 TRPV3 (0.58) PDE10ATRPV3
SCHEMBL29600540 0.73 MAPT (0.41) PIM2KMT2AMEN1CYP3A4CYP2C9
SCHEMBL24324092 0.73 MAPT (0.41) PIM2KMT2AMEN1CYP3A4CYP2C9
SCHEMBL12186828 0.73 CYP1A2 (0.42) PDE10ACYP11B1CYP11B2PIM2KMT2A
SCHEMBL15537503 0.73 TRPV3 (0.57) PDE10ATRPV3SORD
SCHEMBL17221263 0.73 UBE2T (0.40) SORDALDH1A1LMNA
SCHEMBL21875342 0.72 SMN1; SMN2 (0.46) TRPV3KMT2AMEN1CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed