SCHEMBL24326262

SCHEMBL24326262

Cc1cccc(C)c1-c1cc(Cl)nc(NSc2cccc(CN3CCN(C(=O)OC(C)(C)C)C(CC(C)C)C(O)C3)c2)n1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.34
TBK1 Q9UHD2 2/20 0.32
GLS O94925 2/20 0.32
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
JAK1 P23458 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24325795 0.89 TBK1 (0.34) ROCK2TBK1GLS
SCHEMBL24326520 0.87 PARP1 (0.33)
SCHEMBL24326259 0.87 PARP1 (0.33)
SCHEMBL24326675 0.86 MEN1 (0.33)
SCHEMBL24325747 0.86 MEN1 (0.33)
SCHEMBL24326673 0.85 ALDH1A1 (0.40) ROCK2
SCHEMBL24326684 0.82 P2RX3 (0.33) TBK1
SCHEMBL24325771 0.82 GPR119 (0.33) TBK1
SCHEMBL24326190 0.81 TBK1 (0.42) ROCK2TBK1GLSMAPTNPSR1
SCHEMBL24325752 0.79 ALDH1A1 (0.40) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed