SCHEMBL24325771

SCHEMBL24325771

Cc1cccc(C)c1-c1cc(Cl)nc(NSc2cccc(CN3CCCN(C(=O)OC(C)(C)C)CC3CC(C)C)c2)n1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.33
HTR6 P50406 3/20 0.33
TRPV3 Q8NET8 2/20 0.33
USP30 Q70CQ3 1/20 0.33
BCHE P06276 2/20 0.32
BRD4 O60885 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
P2RX3 P56373 2/20 0.32
C5AR1 P21730 1/20 0.32
PARP1 P09874 2/20 0.31
PARP2 Q9UGN5 2/20 0.31
TBK1 Q9UHD2 1/20 0.31
PFKFB3 Q16875 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24325806 0.94 GPR119 (0.34) GPR119HTR6TRPV3USP30BCHE
SCHEMBL24326684 0.91 P2RX3 (0.33) GPR119BRD4P2RX3TBK1
SCHEMBL24326679 0.85 ALDH1A1 (0.41)
SCHEMBL24326190 0.84 TBK1 (0.42) MEN1KMT2APARP1TBK1
SCHEMBL24326719 0.84 GPR119 (0.34) GPR119HTR6TRPV3USP30BCHE
SCHEMBL24325795 0.83 TBK1 (0.34) MEN1KMT2ATBK1
SCHEMBL24326262 0.82 ROCK2 (0.34) TBK1
SCHEMBL24326178 0.80 MMP3 (0.32) TRPV3P2RX3
SCHEMBL24325763 0.80 MMP3 (0.32) TRPV3P2RX3
SCHEMBL24326398 0.79 MEN1 (0.37) TRPV3USP30MEN1KMT2APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed