SCHEMBL2432905

SCHEMBL2432905

Cc1[c]cccc1-c1ccc(F)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.38
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
MAOB P27338 1/20 0.36
CREBBP Q92793 1/20 0.35
STAT3 P40763 1/20 0.35
TNKS O95271 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
NFE2L2 Q16236 1/20 0.34
PTGS2 P35354 4/20 0.34
CD274 Q9NZQ7 1/20 0.34
PTGS1 P23219 1/20 0.33
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
NOTUM Q6P988 1/20 0.33
GLO1 Q04760 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2050955 0.80 PTGS2 (0.36) TGFBR1MAOBCREBBPSTAT3PTGS2
SCHEMBL2013153 0.79 HTR1A (0.35)
SCHEMBL2014605 0.79 PTGS2 (0.42) TGFBR1PTGS2PTGS1
SCHEMBL2012496 0.79 ACHE (0.41) MAOBTNKS2NOTUM
SCHEMBL2428521 0.76 HSD17B1 (0.34) TGFBR1MAOBCREBBPSTAT3ALOX5AP
SCHEMBL6823830 0.76 PTGS2 (0.42) TGFBR1PTGS2PTGS1
SCHEMBL8524724 0.75 AHR (0.47) AKR1C3AKR1C2
SCHEMBL20956991 0.75 ESR2 (0.42)
SCHEMBL2431963 0.75 ACHE (0.34) TGFBR1AKR1C3AKR1C2NFE2L2PTGS2
SCHEMBL2049820 0.75 PTPN1 (0.38) NFE2L2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed