SCHEMBL2437732

SCHEMBL2437732

CCOC(=O)CC(=O)Nc1cc(C(=O)OCC)n[nH]1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.57
NPSR1 Q6W5P4 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TSHR P16473 1/20 0.49
KMT2A Q03164 2/20 0.48
POLB P06746 1/20 0.45
MEN1 O00255 1/20 0.45
HPGD P15428 1/20 0.45
TP53 P04637 1/20 0.42
THRB P10828 1/20 0.42
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14587608 0.84 NPSR1 (0.50) NPSR1L3MBTL1KMT2APOLBHPGD
SCHEMBL13369577 0.81 NPSR1 (0.52) NPSR1L3MBTL1KMT2APOLBTP53
SCHEMBL31001781 0.78 NPSR1 (0.45) NPSR1L3MBTL1KMT2APOLBHPGD
SCHEMBL28563324 0.77 SMN1; SMN2 (0.47) NPSR1L3MBTL1KMT2APOLBHPGD
SCHEMBL25973886 0.77 L3MBTL1 (0.49) NPSR1L3MBTL1KMT2APOLBTP53
SCHEMBL14120046 0.76 PKM (0.51) PKMTSHRKMT2AMEN1HPGD
SCHEMBL23943148 0.75 NPSR1 (0.47) NPSR1L3MBTL1KMT2APOLBTP53
SCHEMBL25312921 0.75 NPSR1 (0.47) NPSR1L3MBTL1KMT2APOLBMEN1
SCHEMBL3825896 0.75 NPSR1 (0.42) NPSR1L3MBTL1KMT2APOLBMEN1
SCHEMBL20746019 0.74 L3MBTL1 (0.58) NPSR1L3MBTL1KMT2APOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250161307-A1 PYRAZOLOPYRIMIDINES AS MODULATORS OF SPERMINE OXIDASE JANSSEN PHARMACEUTICA NV (BE) 2025-05-22 US disclosed
US-12215112-B2 CD151 inhibitors Esfam Biotech Pty Ltd (AU) 2025-02-04 US disclosed
WO-2024254599-A1 HPGD INHIBITORS AND USES THEREOF NIMBUS DISCOVERY, INC. (US) 2024-12-12 WO disclosed
EP-4469454-A1 PYRAZOLOPYRIMIDINES AS MODULATORS OF SPERMINE OXIDASE Janssen Pharmaceutica NV (BE) 2024-12-04 EP disclosed
US-20230365567-A1 COMPOUNDS Esfam Biotech Pty Ltd (AU) 2023-11-16 US disclosed
US-20230365567-A1 COMPOUNDS Esfam Biotech Pty Ltd (AU) 2023-11-16 US disclosed
US-20230365567-A1 COMPOUNDS Esfam Biotech Pty Ltd (AU) 2023-11-16 US disclosed
CN-116829558-A Compounds of formula (I) 艾斯法姆生物技术股份有限公司 2023-09-29 CN disclosed
WO-2023141866-A1 PYRAZOLOPYRIMIDINES AS MODULATORS OF SPERMINE OXIDASE JANSSEN PHARMACEUTICA NV (BE) 2023-08-03 WO disclosed
WO-2023141866-A1 PYRAZOLOPYRIMIDINES AS MODULATORS OF SPERMINE OXIDASE JANSSEN PHARMACEUTICA NV (BE) 2023-08-03 WO disclosed
WO-2022020889-A1 METHOD OF TREATMENT OF CYTOMEGALOVIRUS Esfam Biotech Pty Ltd (AU) 2022-02-03 WO disclosed
WO-2022020891-A1 METHODS OF PROPHYLAXIS AND TREATMENT OF CORONA VIRUS Esfam Biotech Pty Ltd (AU) 2022-02-03 WO disclosed
WO-2022020887-A1 TREATMENT OF CD151 RELATED DISORDERS Esfam Biotech Pty Ltd (AU) 2022-02-03 WO disclosed
WO-2022020888-A1 COMPOUNDS Esfam Biotech Pty Ltd (AU) 2022-02-03 WO disclosed
WO-2022020891-A1 METHODS OF PROPHYLAXIS AND TREATMENT OF CORONA VIRUS Esfam Biotech Pty Ltd (AU) 2022-02-03 WO disclosed
EP-2539342-B1 PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS PDE10 INHIBITORS MITSUBISHI TANABE PHARMA CORP (JP) 2015-04-15 EP disclosed
US-8969376-B2 Pyrazolopyrimidine compounds and their use as PDE10 inhibitors MITSUBISHI TANABE PHARMA CORPORATION (JP) 2015-03-03 US disclosed
EP-2539342-A1 PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS PDE10 INHIBITORS Mitsubishi Tanabe Pharma Corporation (JP) 2013-01-02 EP disclosed
US-20120309754-A1 PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS PDE10 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-12-06 US disclosed
WO-2011105628-A1 PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS PDE10 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-09-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230365567-A1 COMPOUNDS CD81, CD47, CD59 PKM 4516/4885NPSR1 211/4885L3MBTL1 4091/4885
US-12215112-B2 CD151 inhibitors CD81, CD47, CD4 PKM 4831/4885NPSR1 1917/4885L3MBTL1 3502/4885
US-20250161307-A1 PYRAZOLOPYRIMIDINES AS MODULATORS OF SPERMINE OXIDASE SMOX, SRM, SMS PKM 550/4885NPSR1 1352/4885L3MBTL1 1735/4885
US-20120309754-A1 PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS PDE10 INHIBITORS PDE3B, PDE3A, PDE5A PKM 296/4885NPSR1 2131/4885L3MBTL1 4568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.