SCHEMBL24386337

SCHEMBL24386337

O=C(c1ccc(-c2ncon2)cc1)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.44
GPR119 Q8TDV5 1/20 0.40
MAP2K4 P45985 1/20 0.40
MLYCD O95822 8/20 0.39
ACHE P22303 2/20 0.38
HDAC4 P56524 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
HDAC1 Q13547 2/20 0.37
FAAH O00519 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
PIK3CA P42336 1/20 0.36
MTOR P42345 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24386424 0.87 GPR119 (0.39) GPR119HDAC4HDAC6PSEN1PSEN2
SCHEMBL15515155 0.79 TP53 (0.46) GPR119
SCHEMBL19056956 0.75 CES1 (0.65) CES1MAP2K4MLYCDHDAC6HDAC1
SCHEMBL493936 0.75 KIF11 (0.45)
SCHEMBL19976449 0.74 HDAC4 (0.48) MLYCDHDAC4HDAC6HDAC1
SCHEMBL24386409 0.72 GPR119 (0.37) GPR119HDAC6HDAC1
SCHEMBL2740475 0.72 NPC1 (0.40)
SCHEMBL1188116 0.72 MEN1 (0.50)
SCHEMBL15572941 0.71 SCN5A (0.44)
SCHEMBL11712888 0.70 ADORA2A (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3275440-B1 NOVEL OXADIAZOLE DERIVATIVE AND PHARMACEUTICAL CONTAINING SAME NAT CT GERIATRICS & GERONTOLOGY (JP) 2022-05-04 EP disclosed