SCHEMBL244490

SCHEMBL244490

O=C(c1ccc2c(c1)OCCO2)N1CCCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 9/20 1.00
TSHR P16473 2/20 1.00
RECQL P46063 2/20 1.00
CYP1A2 P05177 1/20 0.82
CYP3A4 P08684 1/20 0.82
CYP2D6 P10635 1/20 0.82
CYP2C9 P11712 1/20 0.82
CYP2C19 P33261 1/20 0.82
ALDH1A1 P00352 9/20 0.79
CHRNA7 P36544 1/20 0.73
HSD17B10 Q99714 3/20 0.72
SMN1; SMN2 Q16637 2/20 0.69
PKM P14618 2/20 0.60
MAPT P10636 3/20 0.59
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
GAA P10253 1/20 0.58
LMNA P02545 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14140751 0.90 HPGD (1.00) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL13486221 0.90 HPGD (1.00) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL244547 0.90 HPGD (1.00) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL5970063 0.89 HPGD (1.00) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL14085095 0.84 HPGD (0.73) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL13779946 0.84 HPGD (0.97) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL8475795 0.83 HPGD (0.71) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL13216391 0.83 HPGD (0.71) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL5524809 0.83 HPGD (0.71) HPGDTSHRRECQLCYP1A2CYP3A4
SCHEMBL108225 0.81 ALDH1A1 (0.90) HPGDTSHRRECQLCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 215 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250213564-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALZHEIMER'S DISEASE AND OTHER NEUROGENERATIVE DISEASE THE RESEARCH FOUNDATION FOR MENTAL HYGIENE, INC. 2025-07-03 US claimed
US-20250161264-A1 (AMPAR-PAM)-NMDA RECEPTOR ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF MENTAL CONDITIONS AND DISORDERS GILGAMESH PHARMACEUTICALS, INC. 2025-05-22 US claimed
CN-119504698-A Method for preparing CX546 by using sulfur hexafluoride 国网安徽省电力有限公司电力科学研究院 2025-02-25 CN claimed
US-20250032431-A1 METHODS OF TREATING RETT SYNDROME USING FENFLURAMINE ZOGENIX INTERNATIONAL LIMITED (GB) 2025-01-30 US claimed
US-12144787-B2 Method of treating patients with a mutation in cyclin-dependent kinase-like 5 (CDKL5) ZOGENIX INTERNATIONAL LIMITED (GB) 2024-11-19 US claimed
US-20230285322-A1 Biomarkers for Efficacy of Prophylactic Treatments Against Stress-Induced Affective Disorders THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-09-14 US claimed
WO-2023154450-A2 (AMPA-PAM)-NMDA RECEPTOR ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF MENTAL CONDITIONS AND DISORDERS GILGAMESH PHARMACEUTICALS, INC. (US) 2023-08-17 WO claimed
US-20230142111-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-05-11 US claimed
CN-113932789-B Data transmission method and system for optical fiber gyroscope 宁波圣荣电子科技有限公司 2023-03-07 CN claimed
CN-216012261-U Optical fiber gyroscope 舟山市向海电子科技有限公司 2022-03-11 CN claimed
EP-2948135-B1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS UNIV CASE WESTERN RESERVE (US) 2019-01-02 EP claimed
US-20180008559-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS CASE WESTERN RESERVE UNIVERSITY 2018-01-11 US claimed
US-20170209425-A1 METHODS AND COMPOSITIONS FOR TREATING PATHOLOGIES ASSOCIATED WITH BDNF SIGNALING UNIV CASE WESTERN RESERVE (US) 2017-07-27 US claimed
US-20150359759-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS CASE WESTERN RESERVE UNIVERSITY 2015-12-17 US claimed
EP-2948135-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS Case Western Reserve University (US) 2015-12-02 EP claimed
WO-2014117089-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS CASE WESTERN RESERVE UNIVERSITY (US) 2014-07-31 WO claimed
US-20100035877-A1 METHODS AND COMPOSITIONS FOR TREATING PATHOLOGIES ASSOCIATED WITH BDNF SIGNALING NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR NIH 2010-02-11 US claimed
WO-2008027648-A2 METHODS AND COMPOSITIONS FOR TREATING PATHOLOGIES ASSOCIATED WITH BDNF SIGNALING CASE WESTERN RESERVE UNIVERSITY (US) 2008-03-06 WO claimed
WO-2006034196-A1 COMPOSITIONS FOR ENHANCING MEMORY AND METHODS THEREFOR LIFELIKE BIOMATIC INC. (US) 2006-03-30 WO claimed
US-20060063707-A1 Compositions for enhancing memory and methods therefor LIFELIKE BIOMATIC, INC. (US) 2006-03-23 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063707-A1 Compositions for enhancing memory and methods therefor GRIN1, GRIN3A, GRIN2A HPGD 1202/4885TSHR 3499/4885RECQL 4057/4885
US-20250032431-A1 METHODS OF TREATING RETT SYNDROME USING FENFLURAMINE HTR2C, HTR2A, HTR1A HPGD 3905/4885TSHR 430/4885RECQL 656/4885
US-12144787-B2 Method of treating patients with a mutation in cyclin-dependent kinase-like 5 (CDKL5) CDKL5, HTR5A, CDKL1 HPGD 4022/4885TSHR 1269/4885RECQL 848/4885
US-20230142111-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS GRIN2D, GRIN2A, GRIN2C HPGD 1983/4885TSHR 2725/4885RECQL 4750/4885
US-20170209425-A1 METHODS AND COMPOSITIONS FOR TREATING PATHOLOGIES ASSOCIATED WITH BDNF SIGNALING NTRK2, BDNF, NGF HPGD 3434/4885TSHR 3042/4885RECQL 3635/4885
US-20250161264-A1 (AMPAR-PAM)-NMDA RECEPTOR ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF MENTAL CONDITIONS AND DISORDERS GRIN2A, GRIN1, GRIN3A HPGD 3070/4885TSHR 958/4885RECQL 2820/4885
US-20150359759-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS MECP2, GRIN2A, GRIN2C HPGD 2404/4885TSHR 4233/4885RECQL 3817/4885
US-20180008559-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PERVASIVE DEVELOPMENT DISORDERS GRIN2A, GRIN2C, GRIN2D HPGD 1564/4885TSHR 3490/4885RECQL 4525/4885
US-20100035877-A1 METHODS AND COMPOSITIONS FOR TREATING PATHOLOGIES ASSOCIATED WITH BDNF SIGNALING NTRK2, NGF, BDNF HPGD 2739/4885TSHR 2530/4885RECQL 3458/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.