SCHEMBL24469797

SCHEMBL24469797

Cc1ccnn1-c1ccc(-n2c(=O)c3c(n4ncc(Cc5ccccc5)c24)CN(C(=O)c2ccc(Br)c(Cl)c2)CC3)cc1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
P2RX7 Q99572 2/20 0.33
PDE2A O00408 1/20 0.32
MAPK14 Q16539 3/20 0.31
EEF2K O00418 1/20 0.31
TP53 P04637 2/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
DCTPP1 Q9H773 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
MTHFD2 P13995 1/20 0.31
SPR P35270 1/20 0.30
ITGB2 P05107 1/20 0.30
ICAM1 P05362 1/20 0.30
ITGAL P20701 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24173421 0.91 ALDH1A1 (0.36) ALDH1A1P2RX7TP53MAPTLMNA
SCHEMBL26841996 0.91 P2RX7 (0.33) P2RX7TP53
SCHEMBL26842658 0.90 MAPT (0.35) ALDH1A1P2RX7TP53MAPTLMNA
SCHEMBL24483838 0.89 HDAC1 (0.35) ALDH1A1P2RX7TP53MAPTLMNA
SCHEMBL22845425 0.89 MTHFD2 (0.33) ALDH1A1P2RX7TP53MAPTLMNA
SCHEMBL26842714 0.89 PDE2A (0.34) P2RX7PDE2AEEF2KTP53MAPT
SCHEMBL24469795 0.88 MGLL (0.37) ALDH1A1P2RX7TP53MAPTLMNA
SCHEMBL22845346 0.88 MGLL (0.36) P2RX7PDE2AMAPK14EEF2KTP53
SCHEMBL22845339 0.88 P2RX7 (0.35) ALDH1A1P2RX7MAPTLMNAMTHFD2
SCHEMBL22845445 0.87 MAPT (0.35) ALDH1A1P2RX7TP53MAPTITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11820773-B2 Tricyclic compounds ALIGOS THERAPEUTICS, INC. (US) 2023-11-21 US disclosed
US-11820773-B2 Tricyclic compounds ALIGOS THERAPEUTICS, INC. (US) 2023-11-21 US disclosed
US-20220169650-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2022-06-02 US disclosed
WO-2022115384-A1 TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. (US) 2022-06-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220169650-A1 TRICYCLIC COMPOUNDS SLC10A1, PKD1, CEL ALDH1A1 648/4885P2RX7 2406/4885PDE2A 1720/4885
US-11820773-B2 Tricyclic compounds SLC10A1, PKD1, CEL ALDH1A1 648/4885P2RX7 2406/4885PDE2A 1720/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.