SCHEMBL2448637

SCHEMBL2448637

COc1cc(CC=O)cc(OC)c1Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.42
ERN1 O75460 2/20 0.41
ALDH1A1 P00352 5/20 0.40
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
CA2 P00918 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTGS2 P35354 1/20 0.38
AMY1A P0DUB6 1/20 0.38
CYP3A4 P08684 2/20 0.37
PTGS1 P23219 2/20 0.37
ALOX5 P09917 1/20 0.37
AR P10275 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
MAPT P10636 3/20 0.37
LMNA P02545 2/20 0.37
TNKS O95271 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13403398 0.81 CYP1A2 (0.52) PRKDCALDH1A1CA2TSHRPTGS2
SCHEMBL724406 0.81 PTGS2 (0.59) CA2PTGS2CYP3A4MAPTTUBB1
SCHEMBL4054977 0.79 MAPT (0.51) ERN1CA2KDM4EPTGS2CYP3A4
SCHEMBL30041126 0.78 CA2 (0.43) ALDH1A1PPARGPPARDPPARACA2
SCHEMBL14280291 0.76 ALDH1A1 (0.38) ALDH1A1PPARGPPARDPPARACA2
SCHEMBL15150156 0.76 MEN1 (0.40) ALDH1A1PPARGPPARDPPARACA2
SCHEMBL8429647 0.76 PTGS2 (0.64) ALDH1A1PPARGPPARDPPARACA2
SCHEMBL30644304 0.75 ALDH1A1 (0.69) ALDH1A1PPARGPPARDPPARACA2
SCHEMBL557409 0.75 ALDH1A1 (0.69) ALDH1A1PPARGPPARDPPARACA2
SCHEMBL13403394 0.75 MAPT (0.51) ALDH1A1PPARGPPARDPPARAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2544679-A1 PDE10 INHIBITORS AND RELATED COMPOSITIONS AND METHODS Omeros Corporation (US) 2013-01-16 EP disclosed
WO-2011112828-A1 PDE10 INHIBITORS AND RELATED COMPOSITIONS AND METHODS OMEROS CORPORATION (US) 2011-09-15 WO disclosed