SCHEMBL2452095

SCHEMBL2452095

CC(C)(C)C1(c2ccccc2O)CNCCN1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
HSD17B10 Q99714 2/20 0.32
NPC1 O15118 1/20 0.32
KMT2A Q03164 2/20 0.31
HSD11B1 P28845 1/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRK1 P41145 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
BACE1 P56817 1/20 0.31
PDK2 Q15119 1/20 0.30
RBP4 P02753 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226221 0.73 OPRM1 (0.35) NPC1OPRM1OPRK1SLC6A2SLC6A4
SCHEMBL15094673 0.72 APP (0.39) SIGMAR1HTR2AHTR2CHTR2BHSD17B10
SCHEMBL20362064 0.71 SLC6A2 (0.37) NPC1POLBUSP2PDK2SLC6A2
SCHEMBL3312128 0.68 NPSR1 (0.35) HSD11B1ALDH1A1TSHR
SCHEMBL3313722 0.68 NPSR1 (0.35) HSD11B1ALDH1A1TSHR
SCHEMBL15266847 0.68 RXFP1 (0.40) SIGMAR1HTR2AHTR2CHTR2BHSD17B10
SCHEMBL15094568 0.68 HCAR2 (0.39) SIGMAR1HTR2AHTR2CHTR2BHSD17B10
SCHEMBL3312135 0.68 NPSR1 (0.35) HSD11B1ALDH1A1TSHR
SCHEMBL484224 0.68 HSD17B10 (0.34) HSD17B10NPC1KMT2AMEN1OPRM1
SCHEMBL484225 0.68 HSD17B10 (0.34) HSD17B10NPC1KMT2AMEN1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011112858-A1 PHENOXY THIOPHENE SULFONAMIDES AND THEIR USE AS INHIBITORS OF GLUCURONIDASE NORTH CAROLINA CENTRAL UNIVERSITY (US) 2011-09-15 WO disclosed