SCHEMBL24521975

SCHEMBL24521975

CNc1cccc(CCO)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 4/20 0.50
CYP4A11 Q02928 4/20 0.50
SIRT1 Q96EB6 1/20 0.49
TDP1 Q9NUW8 1/20 0.46
TRPV1 Q8NER1 1/20 0.43
PYGL P06737 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX5 P09917 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
BACE1 P56817 1/20 0.41
HTR6 P50406 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5186512 0.89 CYP4A11 (0.47) CYP4F2CYP4A11SIRT1HTR6GRIN2D
SCHEMBL3150743 0.83 PDK1 (0.49) ALDH1A1MAPTTSHRAPP
SCHEMBL8221872 0.82 GRIN2D (0.51) GAAHTR6GRIN2DGRIN3BGRIN1
Hydrochloric Acid SCHEMBL15823626 0.81 FFAR1 (0.45) CYP4F2CYP4A11ALDH1A1APP
SCHEMBL8283676 0.81 CYP4F2 (0.47) CYP4F2CYP4A11SIRT1TDP1TRPV1
SCHEMBL18905641 0.81 TSHR (0.48) KDM4EMAPTHTR6GRIN2DGRIN3B
SCHEMBL13489892 0.80 ALDH1A1 (0.48) ALDH1A1GAAMAPTHTR6GRIN2D
SCHEMBL6096809 0.80 SIRT1 (0.53) CYP4F2CYP4A11SIRT1TDP1TRPV1
SCHEMBL7401522 0.80 HTR6 (0.43) SIRT1GAAMAPTHTR6GRIN2D
SCHEMBL30046030 0.80 TAAR1 (0.43) HTR6GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4015508-A1 METHODS FOR PREPARING SUBSTITUTED 5,6-DIHYDRO-6-PHENYLBENZO[F]ISOQUINOLIN-2-AMINE ArQule, Inc. (US) 2022-06-22 EP disclosed