SCHEMBL24527435

SCHEMBL24527435

FC(F)(F)c1ccc(N2CCC=N2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.44
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.39
PTGS2 P35354 1/20 0.39
NOTUM Q6P988 2/20 0.38
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
DHFR P00374 1/20 0.37
AKR1C3 P42330 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KIF11 P52732 1/20 0.35
MLYCD O95822 1/20 0.35
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
KDM1A O60341 1/20 0.34
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11401374 0.84 TP53 (0.47) ACHETP53
SCHEMBL17915946 0.81 TP53 (0.43) ACHETP53ALDH1A1KIF11MEN1
SCHEMBL9712169 0.80 ALOX5 (0.56) PTGS2NOTUMKDM4EALDH1A1TSHR
SCHEMBL30720446 0.76 DHFR (0.44) ACHETP53CYP3A4DHFRHRH3
SCHEMBL981604 0.75 TP53 (0.42) TP53NOTUMKDM4EALDH1A1
SCHEMBL11027181 0.75 TP53 (0.42) ACHETP53TDP1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL28999664 0.73 TP53 (0.41) TP53NOTUMAKR1C3KDM4EALDH1A1
SCHEMBL28229221 0.70 NOTUM (0.38) CYP3A4PTGS2NOTUMCA12CA2
SCHEMBL29222359 0.69 TP53 (0.55) TP53CA12CA2TDP1KDM4E
SCHEMBL28650484 0.69 CA12 (0.65) CYP3A4NOTUMCA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022132803-A1 CB2 RECEPTOR AGONISTS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2022-06-23 WO disclosed
WO-2022132803-A1 CB2 RECEPTOR AGONISTS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2022-06-23 WO disclosed