SCHEMBL2453353

SCHEMBL2453353

CCCCOC(=O)N1CCC(c2cscc2C(=O)OC)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
KDM4E B2RXH2 2/20 0.41
MMP13 P45452 2/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HTT P42858 2/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
EED O75530 1/20 0.37
RBBP4 Q09028 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2447286 0.82 POLB (0.44) SMN1; SMN2LMNAPOLBMMP13MMP2
SCHEMBL2419233 0.80 RBP4 (0.41) SMN1; SMN2LMNAKDM4ECHRM2CHRM1
SCHEMBL2428188 0.79 EED (0.54) POLBKDM4EALDH1A1HTTEED
SCHEMBL2454067 0.79 ALDH1A1 (0.43) SMN1; SMN2LMNAPOLBKDM4EMMP13
SCHEMBL2454613 0.79 LMNA (0.41) SMN1; SMN2LMNAPOLBKDM4EMMP13
SCHEMBL2454973 0.77 CHRM2 (0.45) SMN1; SMN2LMNAPOLBKDM4EMMP13
SCHEMBL2444427 0.77 LMNA (0.44) SMN1; SMN2LMNAPOLBKDM4EMMP13
SCHEMBL2278659 0.74 TSHR (0.46) SMN1; SMN2LMNAPOLBALDH1A1GAA
SCHEMBL2446770 0.73 FABP6 (0.38) SMN1; SMN2LMNAPOLBKDM4ECYP1A2
SCHEMBL28225300 0.72 BRD4 (0.57) SMN1; SMN2LMNAPOLBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2550252-A1 1-(2-PHENOXYMETHYLHETEROARYL)PIPERIDINE AND PIPERAZINE COMPOUNDS Theravance, Inc. (US) 2013-01-30 EP disclosed
WO-2011119461-A1 1-(2-PHENOXYMETHYLHETEROARYL)PIPERIDINE AND PIPERAZINE COMPOUNDS THERAVANCE, INC. (US) 2011-09-29 WO disclosed