SCHEMBL24566902

SCHEMBL24566902

C[Si](C)(C)CCOCn1nc(C2CC2)c2cc(Br)cnc21

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.36
KLKB1 P03952 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29705582 1.00 DGAT1 (0.36) DGAT1KLKB1
SCHEMBL27215183 0.86 KLKB1 (0.33) DGAT1KLKB1
SCHEMBL30592405 0.85 MTNR1A (0.36) DGAT1KLKB1
SCHEMBL3300284 0.83 DGAT1 (0.39) DGAT1
SCHEMBL27215111 0.82 DGAT1 (0.38) DGAT1
SCHEMBL1593371 0.82 DGAT1 (0.38) DGAT1
SCHEMBL27193468 0.81 DGAT1 (0.37) DGAT1
SCHEMBL27193478 0.80 DGAT1 (0.37) DGAT1
SCHEMBL24566116 0.80 DGAT1 (0.37) DGAT1
SCHEMBL24566903 0.80 GSK3A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250221988-A1 COMPOUNDS AND METHODS OF TREATING CANCERS CULLGEN (SHANGHAI), INC. (CN) 2025-07-10 US disclosed
US-20240150345-A1 GCN2 MODULATING COMPOUNDS AND USES THEREOF PHARMARON UK LTD. (GB) 2024-05-09 US disclosed
WO-2022140527-A1 6-HETEROARYLOXY BENZIMIDAZOLES AND AZABENZIMIDAZOLES AS JAK2 INHIBITORS AJAX THERAPEUTICS, INC. (US) 2022-06-30 WO disclosed
CN-103214480-B Pyrazolopyridine alkynes benzene-like compounds and medicinal compositions thereof and application GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2015-12-16 CN disclosed
CN-103214480-A Pyrazolopyridines alkynylbenzene compound and medicinal composition and application GUANGZHOU INST BIOMED & HEALTH 2013-07-24 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250221988-A1 COMPOUNDS AND METHODS OF TREATING CANCERS GSPT1, GSS, G6PC1 DGAT1 206/4885KLKB1 713/4885
US-20240150345-A1 GCN2 MODULATING COMPOUNDS AND USES THEREOF EIF2AK4, GCN1, CLN6 DGAT1 565/4885KLKB1 4832/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.