SCHEMBL2461969

SCHEMBL2461969

Cc1[nH]c2nc(N)nn2c(=O)c1Cc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 1/20 0.39
TLR7 Q9NYK1 3/20 0.38
TBXAS1 P24557 2/20 0.38
GFER P55789 1/20 0.37
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK1 P06493 1/20 0.37
CDK4 P11802 1/20 0.37
CCNB1 P14635 1/20 0.37
CCND1 P24385 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2462018 0.86 PDE10A (0.40) PNPTLR7TBXAS1CCNB2CCNE2
SCHEMBL2454543 0.81 ADCY10 (0.44) KDM4EALDH1A1HPGD
SCHEMBL2459259 0.81 CCR2 (0.51) PNP
SCHEMBL2464343 0.80 ALKBH3 (0.40) CCNE2CCNE1CDK2KDM4EALDH1A1
SCHEMBL12324736 0.78 CCR2 (0.46)
SCHEMBL12325085 0.78 NPSR1 (0.48) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL12324671 0.78 PARP14 (0.42) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL2457171 0.77 ALKBH3 (0.48) PNPMEN1KMT2AALDH1A1HPGD
SCHEMBL12324675 0.76 KDM4E (0.40) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL2461272 0.75 ALKBH3 (0.38) KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114148-A1 4H- [1, 2, 4] TRIAZOLO [5, 1 -B] PYRIMIDIN-7 -ONE DERIVATIVES AS CCR2B RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2011-09-22 WO claimed
WO-2011114148-A1 4H- [1, 2, 4] TRIAZOLO [5, 1 -B] PYRIMIDIN-7 -ONE DERIVATIVES AS CCR2B RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2011-09-22 WO disclosed
WO-2011114148-A1 4H- [1, 2, 4] TRIAZOLO [5, 1 -B] PYRIMIDIN-7 -ONE DERIVATIVES AS CCR2B RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2011-09-22 WO disclosed