SCHEMBL2464168

SCHEMBL2464168

CCCOc1cc2c(c3c(=O)c(-c4ccc(OC)cc4)cn(OC(C)=O)c13)C(CC)CCO2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.35
ESR2 Q92731 3/20 0.35
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
EDNRA P25101 3/20 0.33
EDNRB P24530 2/20 0.33
LTB4R Q15722 1/20 0.32
LTB4R2 Q9NPC1 1/20 0.32
TERT O14746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362491 0.83 ESR1 (0.38) ESR1ESR2CNR1CNR2MTNR1A
SCHEMBL2461978 0.76 CHRM1 (0.40) CNR1CNR2MTNR1AMTNR1BKDM4E
SCHEMBL2578644 0.69 ESR1 (0.42) ESR1ESR2CNR1CNR2KDM4E
SCHEMBL2464167 0.68 ESR1 (0.34) ESR1ESR2MTNR1AMTNR1BKDM4E
SCHEMBL2581042 0.68 ESR1 (0.37) ESR1ESR2CNR1CNR2KDM4E
SCHEMBL7910678 0.68 RAB9A (0.40) ESR1ESR2CNR1CNR2
SCHEMBL2460915 0.67 MGAM (0.34) KDM4E
SCHEMBL2586745 0.67 ESR1 (0.36) ESR1ESR2CNR1CNR2
SCHEMBL12160478 0.66 ESR1 (0.38) ESR1ESR2CNR1CNR2EDNRA
SCHEMBL2586818 0.65 ESR1 (0.34) ESR1ESR2CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364298-A1 Quinolone compound and pharmaceutical composition Otsuka Pharmaceutical Co., Ltd. (JP) 2011-09-14 EP disclosed