SCHEMBL2464167

SCHEMBL2464167

CCCOc1cc2c(c3c(=O)c(-c4ccc(OC)cc4)c(CC)n(OC(C)=O)c13)CCCO2

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.34
ESR2 Q92731 3/20 0.34
PTGS2 P35354 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
FPR1 P21462 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
TERT O14746 1/20 0.33
BRD4 O60885 1/20 0.32
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
GRIA2 P42262 1/20 0.31
GRIA4 P48058 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362491 0.83 ESR1 (0.38) ESR1ESR2MTNR1AMTNR1BRAB9A
SCHEMBL2489539 0.78 CHRM1 (0.37) PTGS2MTNR1AMTNR1BFPR1KDM4E
SCHEMBL2578644 0.76 ESR1 (0.42) ESR1ESR2PTGS2RAB9AKDM4E
SCHEMBL2581042 0.75 ESR1 (0.37) ESR1ESR2PTGS2RAB9AKDM4E
SCHEMBL7910678 0.74 RAB9A (0.40) ESR1ESR2RAB9AMAPTMEN1
SCHEMBL2586745 0.73 ESR1 (0.36) ESR1ESR2RAB9A
SCHEMBL2586818 0.72 ESR1 (0.34) ESR1ESR2
SCHEMBL2464402 0.71 ESR1 (0.33) ESR1ESR2
SCHEMBL2581768 0.71 ALDH1A1 (0.35) ESR1ESR2RAB9AKDM4EMAPT
SCHEMBL12175815 0.70 ESR1 (0.31) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364298-A1 Quinolone compound and pharmaceutical composition Otsuka Pharmaceutical Co., Ltd. (JP) 2011-09-14 EP disclosed