SCHEMBL2464560

SCHEMBL2464560

Cc1cc(N)cc(Cl)c1CC=O

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.39
ALDH1A1 P00352 3/20 0.37
THRB P10828 1/20 0.34
IMPDH2 P12268 2/20 0.34
CD44 P16070 1/20 0.33
TSHR P16473 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467191 0.86 ALDH1A1 (0.36) ALDH1A1IMPDH2TSHR
SCHEMBL14992608 0.78 IMPDH2 (0.32) ALDH1A1IMPDH2TSHR
SCHEMBL2464673 0.78 IMPDH2 (0.31) IMPDH2
SCHEMBL2464817 0.74 P2RX7 (0.33) ALDH1A1TSHR
SCHEMBL17182454 0.73 CYP3A4 (0.42) CYP3A4ALDH1A1THRBCD44TSHR
SCHEMBL525350 0.71 CYP3A4 (0.65) CYP3A4ALDH1A1THRBCD44TSHR
SCHEMBL23507137 0.69 P2RX7 (0.40) ALDH1A1
SCHEMBL6155985 0.69 CD44 (0.35) CYP3A4ALDH1A1CD44TSHR
SCHEMBL9566566 0.69 ALDH1A1 (0.46) CYP3A4ALDH1A1THRBTSHR
SCHEMBL1124861 0.69 HRH3 (0.36) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2785714-A1 IMPROVED MODULATORS OF HEC1 ACTIVITY AND METHODS THEREFOR Taivex Therapeutics Corporation (TW) 2014-10-08 EP disclosed
WO-2013082324-A1 IMPROVED MODULATORS OF HEC1 ACTIVITY AND METHODS THEREFOR TAIVEX THERAPEUTICS CORPORATION (TW) 2013-06-06 WO disclosed
EP-2547676-A2 MODULATORS OF HEC1 ACTIVITY AND METHODS THEREFOR Taivex Therapeutics Inc. (TW) 2013-01-23 EP disclosed
WO-2011115998-A2 MODULATORS OF HEC1 ACTIVITY AND METHODS THEREFOR TAIVEX THERAPEUTICS INC. (CN) 2011-09-22 WO disclosed