SCHEMBL2464938

SCHEMBL2464938

COc1ccc([C@H](C)NC(=O)CC(C)=O)cc1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.63
ACACB O00763 2/20 0.60
KMT2A Q03164 3/20 0.57
MEN1 O00255 2/20 0.57
GAA P10253 1/20 0.57
CNR1 P21554 4/20 0.53
KDM4E B2RXH2 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
GPR139 Q6DWJ6 3/20 0.49
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
CNR2 P34972 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464936 1.00 ALDH1A1 (0.63) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL29151019 0.85 ALDH1A1 (0.65) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL15918472 0.85 CNR1 (0.68) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL13683332 0.84 ALDH1A1 (0.63) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL7714868 0.84 ALDH1A1 (0.63) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL23122976 0.84 ALDH1A1 (0.68) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL13898948 0.84 ALDH1A1 (0.63) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL23122978 0.84 ALDH1A1 (0.68) ALDH1A1ACACBKMT2AMEN1GAA
SCHEMBL4446314 0.83 ACACB (0.82) ALDH1A1ACACBKMT2AMEN1CNR1
SCHEMBL4446311 0.83 ACACB (0.82) ALDH1A1ACACBKMT2AMEN1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022218-B2 Hypogonadism; N-{3-[2-Bromo-4-(3-cyano-2-methyl-5-oxo-7-propyl-1,4,5,6,7,8-hexahydro-quinolin-4-yl)-6-ethoxy-phenoxymethyl]-phenyl}-3,4,5-trimethoxy-benzamide; low molecular weight hormone mimetics; selective Follicle Stimulating Hormone receptor agonists N.V. ORGANON (NL) 2011-09-20 US disclosed
US-20080275042-A1 4-Phenyl-5-Oxo-1,4,5,6,7,8-Hexahydroquinoline Derivatives for the Treatment of Infertility N.V. ORGANON (NL) 2008-11-06 US disclosed
EP-1881830-B1 4-PHENYL-5-OXO-1,4,5,6,7,8-HEXAHYDROQUINOLINE DERIVATIVES THE TREATMENT OF INFERTILITY ORGANON NV (NL) 2008-10-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080275042-A1 4-Phenyl-5-Oxo-1,4,5,6,7,8-Hexahydroquinoline Derivatives for the Treatment of Infertility CATSPER1, ABCB11, ACR ALDH1A1 79/4885ACACB 1538/4885KMT2A 1161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.