SCHEMBL2465152

SCHEMBL2465152

C[Si](C)(C)C#Cc1ccc(N(N)C(=O)O)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.35
GABRG2 P18507 5/20 0.35
GABRB3 P28472 5/20 0.35
GABRA5 P31644 5/20 0.35
GABRA3 P34903 5/20 0.35
GABRA2 P47869 5/20 0.35
APP P05067 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
FFAR1 O14842 1/20 0.33
GABRA6 Q16445 3/20 0.32
GABRA4 P48169 2/20 0.32
ADK P55263 2/20 0.31
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
CYP2C19 P33261 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2138873 0.79 GABRA1 (0.42) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11512104 0.77 NPSR1 (0.42) NPSR1MEN1ALDH1A1HPGDCYP2C19
SCHEMBL2465630 0.76 MEN1 (0.30) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6851297 0.75 GABRA1 (0.33) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6036758 0.74 RARB (0.55) ALDH1A1HPGDCYP3A4TSHRRARB
SCHEMBL1306384 0.74 GABRA1 (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL18526935 0.74 ALDH1A1 (0.48) APPADKALDH1A1CYP3A4MAPT
SCHEMBL25093690 0.73 NOS1 (0.44) ALDH1A1CYP2C19KMT2ACYP3A4MAPT
SCHEMBL14882956 0.73 ALDH1A1 (0.42) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1306505 0.72 APP (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367599-A1 INHIBITION OF HDAC2 TO PROMOTE MEMORY Massachusetts Institute of Technology (US) 2011-09-28 EP disclosed
WO-2010065117-A1 INHIBITION OF HDAC2 TO PROMOTE MEMORY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-06-10 WO disclosed