SCHEMBL2465978

SCHEMBL2465978

COC(=O)Oc1nc(-c2ccc(Cl)c(OC)c2F)cc(NC(C)=O)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
ADORA3 P0DMS8 5/20 0.37
TAS1R3 Q7RTX0 2/20 0.37
TAS1R1 Q7RTX1 2/20 0.37
TAS1R2 Q8TE23 2/20 0.37
ADORA2A P29274 4/20 0.36
ADORA2B P29275 2/20 0.36
MEP1B Q16820 1/20 0.35
ABL1 P00519 1/20 0.35
ADORA1 P30542 1/20 0.35
TSHR P16473 1/20 0.34
NUDT1 P36639 1/20 0.34
PDCD1LG2 Q9BQ51 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
RIPK1 Q13546 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2469725 0.92 ALDH1A1 (0.40) ALDH1A1ADORA3TAS1R3TAS1R1TAS1R2
SCHEMBL2468173 0.91 ADORA2A (0.39) ALDH1A1ADORA3ADORA2AADORA2BABL1
SCHEMBL17797223 0.91 RORC (0.40) ALDH1A1ADORA3TAS1R3TAS1R1ABL1
SCHEMBL2468120 0.91 ALDH1A1 (0.36) ALDH1A1ADORA3ADORA2AABL1ADORA1
SCHEMBL2468304 0.89 ALDH1A1 (0.38) ALDH1A1ADORA3ADORA2AABL1ADORA1
SCHEMBL2470796 0.89 ALDH1A1 (0.35) ALDH1A1ADORA3ADORA2AABL1ADORA1
SCHEMBL2464613 0.88 ADORA2A (0.39) ALDH1A1ADORA3ADORA2AADORA2BABL1
SCHEMBL17797221 0.88 TMPRSS4 (0.36) ADORA3ADORA2AADORA2BPDCD1LG2CD274
SCHEMBL3454141 0.87 POLB (0.39) ALDH1A1ADORA3ADORA2AABL1ADORA1
SCHEMBL2468807 0.87 MEP1B (0.36) ALDH1A1TAS1R3TAS1R1TAS1R2MEP1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2797932-B1 METHODS OF ISOLATING (4-CHLORO-2-FLUORO-3-SUBSTITUTED-PHENYL) BORONATES AND METHODS OF USING THE SAME DOW AGROSCIENCES LLC (US) 2017-02-01 EP claimed
EP-2797890-B1 METHODS OF PRODUCING METHYL 4-AMINO-3-CHLORO-6-(4-CHLORO-2-FLUORO-3-METHOXYPHENYL)PYRIDINE-2-CARBOXYLATE DOW AGROSCIENCES LLC (US) 2016-10-05 EP claimed
EP-2060566-B1 Poly-substituted aryls DOW AGROSCIENCES LLC (US) 2016-06-08 EP claimed
EP-2939541-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2369929-A2 HERBICIDE-SAFENER COMBINATION Bayer CropScience AG (DE) 2011-10-05 EP disclosed
WO-2010060581-A2 HERBICIDE-SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 WO disclosed
EP-2191719-A1 Herbicide safener combination Bayer CropScience AG (DE) 2010-06-02 EP disclosed