SCHEMBL2469725

SCHEMBL2469725

COC(=O)Oc1nc(-c2ccc(Cl)c(OC)c2Cl)cc(NC(C)=O)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
ADORA3 P0DMS8 6/20 0.38
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
NUDT1 P36639 1/20 0.38
TSHR P16473 1/20 0.36
ALPL P05186 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
PDCD1LG2 Q9BQ51 4/20 0.35
CD274 Q9NZQ7 4/20 0.35
SCN9A Q15858 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN3A Q9NY46 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2465978 0.92 ALDH1A1 (0.38) ALDH1A1ADORA3ADORA2AADORA2BNUDT1
SCHEMBL2464613 0.89 ADORA2A (0.39) ALDH1A1ADORA3ADORA2AADORA2BNUDT1
SCHEMBL2464008 0.88 NUDT1 (0.41) ALDH1A1ADORA3NUDT1ALPLPDCD1LG2
SCHEMBL17797246 0.86 ALDH1A1 (0.36) ALDH1A1ADORA3NUDT1ALPLPDCD1LG2
SCHEMBL2468173 0.85 ADORA2A (0.39) ALDH1A1ADORA3ADORA2AADORA2BPDCD1LG2
SCHEMBL2470012 0.85 ALDH1A1 (0.38) ALDH1A1ADORA3NUDT1ALPLPDCD1LG2
SCHEMBL17797223 0.85 RORC (0.40) ALDH1A1ADORA3TAS1R3TAS1R1
SCHEMBL2468120 0.85 ALDH1A1 (0.36) ALDH1A1ADORA3ADORA2ANUDT1SCN9A
SCHEMBL2470407 0.85 PDCD1LG2 (0.38) ALDH1A1ALPLPDCD1LG2CD274SCN9A
SCHEMBL17797205 0.84 ALDH1A1 (0.38) ALDH1A1ADORA3NUDT1ALPLPDCD1LG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060566-B1 Poly-substituted aryls DOW AGROSCIENCES LLC (US) 2016-06-08 EP claimed
EP-2939540-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2939541-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2369929-A2 HERBICIDE-SAFENER COMBINATION Bayer CropScience AG (DE) 2011-10-05 EP disclosed
WO-2010060581-A2 HERBICIDE-SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 WO disclosed
EP-2191719-A1 Herbicide safener combination Bayer CropScience AG (DE) 2010-06-02 EP disclosed