SCHEMBL24670463

SCHEMBL24670463

C=C(N)N1CC=C(c2ncc(C(=O)Nc3ccc(CNC(=N)N)cc3)s2)CC1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.40
PTPN1 P18031 1/20 0.39
ROCK2 O75116 2/20 0.38
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
TRPV1 Q8NER1 7/20 0.36
PPARA Q07869 1/20 0.35
EGLN1 Q9GZT9 1/20 0.34
WNT3A P56704 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
NAMPT P43490 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29802997 0.93 PTPN11 (0.39) PTPN11PTPN1ROCK2SLC6A3KCNH2
SCHEMBL24671076 0.84 PTPN11 (0.38) PTPN11PTPN1SLC6A3KCNH2TAAR1
SCHEMBL24670475 0.80 PTPN11 (0.46) PTPN11PTPN1MAPTNAMPT
Trifluoroacetic Acid SCHEMBL29803396 0.80 TRPV1 (0.38) PTPN11PTPN1TRPV1EGLN1WNT3A
SCHEMBL24671549 0.78 TP53 (0.40) PTPN11ROCK2TP53MAPT
SCHEMBL24671535 0.77 TMPRSS2 (0.39) TRPV1EGLN1TP53MAPTJAK2
SCHEMBL29803758 0.77 NAMPT (0.48) WNT3AMAPTNAMPT
SCHEMBL24669641 0.76 EGLN1 (0.41) EGLN1MAPTJAK2JAK1NAMPT
SCHEMBL24669239 0.75 MMP12 (0.38) EGLN1TP53MAPTNAMPT
Trifluoroacetic Acid SCHEMBL29803352 0.75 PTPN11 (0.43) PTPN11PTPN1TRPV1EGLN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed