SCHEMBL24671577

SCHEMBL24671577

COc1cc(C2=CCN(C(=N)N)CC2)ccc1C(=O)Nc1ccc(C2=CCN(C(=N)N)CC2)cn1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.47
NPC1 O15118 5/20 0.47
RAB9A P51151 5/20 0.47
MITF O75030 2/20 0.47
TP53 P04637 1/20 0.47
GAA P10253 1/20 0.47
QDPR P09417 1/20 0.47
NAMPT P43490 9/20 0.45
ABCC1 P33527 2/20 0.44
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 2/20 0.42
RXFP1 Q9HBX9 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24669665 0.86 NAMPT (0.48) ABCB1NPC1RAB9AMITFTP53
SCHEMBL24670310 0.80 PDE4B (0.43) ABCB1NPC1RAB9AMITFTP53
SCHEMBL29803430 0.79 NAMPT (0.44) ABCB1NPC1RAB9AMITFTP53
SCHEMBL24671576 0.79 NAMPT (0.44) ABCB1NPC1RAB9AMITFTP53
SCHEMBL24670528 0.79 NAMPT (0.46) NPC1RAB9ANAMPT
SCHEMBL29802891 0.78 APOBEC3A (0.49) RAB9AQDPRNAMPTKDM4EKMT2A
SCHEMBL29803621 0.77 QDPR (0.54) ABCB1NPC1RAB9AMITFTP53
SCHEMBL24671431 0.76 NAMPT (0.48) NAMPT
SCHEMBL24670801 0.75 TMPRSS2 (0.45) QDPRNAMPTKDM4EKMT2A
SCHEMBL24671261 0.74 QDPR (0.43) ABCB1NPC1RAB9AQDPRNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO claimed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed