SCHEMBL24673381

SCHEMBL24673381

CCc1cccc2c1C(=O)C(=O)NC2=O

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 12/20 0.51
CASP2 P42575 2/20 0.48
CASP7 P55210 2/20 0.48
CASP6 P55212 2/20 0.48
CASP8 Q14790 2/20 0.48
GSK3B P49841 1/20 0.45
PDK2 Q15119 2/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PARP1 P09874 1/20 0.42
DAO P14920 1/20 0.42
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2408327 0.89 KDM4E (0.49) CASP3CASP2CASP7CASP6CASP8
SCHEMBL10883505 0.80 MAOA (0.48) PDK2ALDH1A1HPGDHSD17B10CYP2D6
SCHEMBL8194264 0.80 KDM4E (0.42) CASP3CASP2CASP7CASP6CASP8
SCHEMBL1871243 0.79 CES1 (0.56) CASP3GSK3BPDK2KDM4EDAO
Vinyl Chloride SCHEMBL28309108 0.78 KDM4E (0.41) CASP3CASP2CASP7CASP6CASP8
SCHEMBL9980565 0.77 KDM4E (0.43) CASP3CASP2CASP7CASP6CASP8
SCHEMBL22525286 0.77 DAO (0.58) CASP3CASP2CASP7CASP6CASP8
SCHEMBL1892075 0.76 KDM4E (0.45) CASP3CASP2CASP7CASP6CASP8
SCHEMBL28045932 0.76 GABRA1 (0.43) GSK3BPDK2PARP1DAOCYP2D6
SCHEMBL18983060 0.76 MAPT (0.46) PDK2ALDH1A1HPGDHSD17B10CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230149549-A1 SMARCA DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2023-05-18 US disclosed
US-20230135894-A1 MK2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2023-05-04 US disclosed
US-20220340570-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2022-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230135894-A1 MK2 DEGRADERS AND USES THEREOF MKNK2, MKRN3, DUS2 CASP3 4069/4885CASP2 873/4885CASP7 3628/4885
US-20230149549-A1 SMARCA DEGRADERS AND USES THEREOF SMARCA1, SMARCB1, SMARCE1 CASP3 4064/4885CASP2 3809/4885CASP7 3993/4885
US-20220340570-A1 IRAK DEGRADERS AND USES THEREOF IRAK2, IRAK3, IRAK1 CASP3 816/4885CASP2 406/4885CASP7 456/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.