SCHEMBL24674845

SCHEMBL24674845

CCOC(=O)COc1cccc(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.56
PPARG P37231 1/20 0.56
BRD4 O60885 1/20 0.46
PPID Q08752 1/20 0.44
GLS O94925 2/20 0.44
ROCK2 O75116 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ROCK1 Q13464 1/20 0.43
MMP13 P45452 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19387601 0.84 KDM4E (0.45) PPARAPPARGROCK2
SCHEMBL7475639 0.82 SMN1; SMN2 (0.56) PPARAPPARGCYP3A4CYP2C9SMN1; SMN2
SCHEMBL18705329 0.81 ALDH1A1 (0.46) PPARAPPARGSMN1; SMN2
SCHEMBL1669761 0.81 NAMPT (0.41) PPARAPPARGCYP3A4CYP2D6SMN1; SMN2
SCHEMBL10799448 0.81 PPARA (0.55) PPARAPPARGSMN1; SMN2
SCHEMBL14431530 0.81 PPARA (0.57) PPARAPPARG
SCHEMBL24674846 0.81 ROCK2 (0.47) BRD4GLSROCK2CYP3A4CYP2D6
SCHEMBL3418637 0.80 ALDH1A1 (0.62) MMP13SMN1; SMN2
SCHEMBL24674847 0.80 GLS (0.46) BRD4GLSMMP13SMN1; SMN2
SCHEMBL23461821 0.80 ROCK2 (0.49) BRD4GLSROCK2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022159688-A1 DEGRADERS OF GRK2 AND USES THEREOF CYGNAL THERAPEUTICS, INC. (US) 2022-07-28 WO disclosed