SCHEMBL2467530

SCHEMBL2467530

Nc1cc(-c2ccccc2F)nc(OC(=O)O)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.40
ADORA1 P30542 6/20 0.40
ADORA3 P0DMS8 4/20 0.40
ADORA2B P29275 1/20 0.40
ATR Q13535 1/20 0.39
MPL P40238 1/20 0.38
VCP P55072 1/20 0.36
PARP1 P09874 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
LTB4R Q15722 2/20 0.36
TACR3 P29371 1/20 0.36
NPC1 O15118 1/20 0.35
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464096 0.87 HSP90AA1 (0.46) ADORA2AADORA1ATRVCPKDM5B
SCHEMBL2466888 0.86 KMO (0.43) NPC1
SCHEMBL2468072 0.86 KMO (0.47) PIM3
SCHEMBL2465208 0.86 PIM1 (0.34) PIM1PIM3PIM2
SCHEMBL2469200 0.85 PRKDC (0.39) ADORA2AADORA1ATRVCPTACR3
SCHEMBL2464666 0.84 GRM2 (0.40)
SCHEMBL2470000 0.84 ACHE (0.45) ADORA2AADORA1ADORA3
SCHEMBL2469711 0.84 CYP3A4 (0.34)
SCHEMBL2468802 0.82 HSP90AA1 (0.52) ADORA2AADORA1ADORA3ATRVCP
SCHEMBL2466413 0.81 GRM2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2939540-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2939541-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2369929-A2 HERBICIDE-SAFENER COMBINATION Bayer CropScience AG (DE) 2011-10-05 EP disclosed
WO-2010060581-A2 HERBICIDE-SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 WO disclosed
EP-2191719-A1 Herbicide safener combination Bayer CropScience AG (DE) 2010-06-02 EP disclosed