SCHEMBL2469711

SCHEMBL2469711

Nc1cc(-c2ccc(F)c(F)c2F)nc(OC(=O)O)c1Cl

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.34
KMO O15229 2/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
PDCD1LG2 Q9BQ51 2/20 0.33
CD274 Q9NZQ7 2/20 0.33
GRM2 Q14416 2/20 0.32
GRIN2B Q13224 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3455298 0.89 GRIN2B (0.34) CYP3A4KMOPDCD1LG2CD274GRM2
SCHEMBL17797218 0.88 PDCD1LG2 (0.37) PDCD1LG2CD274
SCHEMBL2468072 0.88 KMO (0.47) CYP3A4KMOGRM2GRIN2B
SCHEMBL2470061 0.87 PDCD1LG2 (0.35) PDCD1LG2CD274
SCHEMBL17797209 0.85 MAPK9 (0.37) KMOPDCD1LG2CD274FFAR4
SCHEMBL2466888 0.85 KMO (0.43) KMOKEAP1GRM2
SCHEMBL17797261 0.84 PDCD1LG2 (0.40) CYP3A4KMOPDCD1LG2CD274
SCHEMBL2469850 0.84 PPARA (0.33) KMOFFAR4
SCHEMBL2467541 0.84 ALDH1A1 (0.37) PDCD1LG2CD274FFAR4
SCHEMBL2467530 0.84 ADORA2A (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060566-B1 Poly-substituted aryls DOW AGROSCIENCES LLC (US) 2016-06-08 EP claimed
EP-2939540-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2939541-A1 HERBICIDE SAFENER COMBINATION Bayer Intellectual Property GmbH (DE) 2015-11-04 EP disclosed
EP-2369929-A2 HERBICIDE-SAFENER COMBINATION Bayer CropScience AG (DE) 2011-10-05 EP disclosed
WO-2010060581-A2 HERBICIDE-SAFENER COMBINATION BAYER CROPSCIENCE AG (DE) 2010-06-03 WO disclosed
EP-2191719-A1 Herbicide safener combination Bayer CropScience AG (DE) 2010-06-02 EP disclosed