SCHEMBL24676993

SCHEMBL24676993

FC(F)(F)c1csc([C@]2(F)C[C@H](OCc3ccccc3)C2)n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.36
OPRL1 P41146 2/20 0.36
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSK P43235 1/20 0.34
DPP4 P27487 1/20 0.34
TACR1 P25103 8/20 0.33
DRD4 P21917 4/20 0.32
SIGMAR1 Q99720 4/20 0.32
KCNH2 Q12809 1/20 0.32
DRD3 P35462 1/20 0.32
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754918 1.00 OPRM1 (0.36) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL29754893 0.87 OPRM1 (0.36) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL24676757 0.87 OPRM1 (0.36) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL24676864 0.77 TACR1 (0.33) CTSKTACR1KCNH2
SCHEMBL24676758 0.76 TRPV1 (0.37) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL25025800 0.75 P2RX7 (0.38) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL20284996 0.72 OPRM1 (0.51) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL29754940 0.70 OPRM1 (0.32) OPRM1OPRL1
SCHEMBL3830852 0.70 CTSL (0.49) OPRM1OPRL1CTSLCTSBCTSK
SCHEMBL446380 0.68 CTSL (0.39) OPRM1OPRL1CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed