SCHEMBL24677400

SCHEMBL24677400

O=CNCc1ccc(CN2CCNCC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 13/20 0.56
SIGMAR1 Q99720 1/20 0.54
MEN1 O00255 1/20 0.54
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
ADRA2C P18825 1/20 0.54
CCR2 P41597 1/20 0.54
CXCL12 P48061 1/20 0.54
BLM P54132 1/20 0.54
KMT2A Q03164 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
HRH3 Q9Y5N1 1/20 0.54
ADH1B P00325 1/20 0.46
ADH1C P00326 1/20 0.46
ADH1A P07327 1/20 0.46
ADH7 P40394 1/20 0.46
CRBN Q96SW2 1/20 0.44
NCF1 P14598 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076451 0.81 CXCR4 (0.67) CXCR4SIGMAR1MEN1CHRM2CHRM1
SCHEMBL5990981 0.81 HRH3 (0.59) HRH3
SCHEMBL12503437 0.81 LMNA (0.56) HRH3ADH1BADH1CADH1AADH7
SCHEMBL24677480 0.81 ADRB1 (0.47) SIGMAR1ADH1BADH1CADH1AADH7
SCHEMBL1259387 0.78 CXCR4 (0.81) CXCR4SIGMAR1MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL5573232 0.78 CXCR4 (0.78) CXCR4SIGMAR1MEN1CHRM2CHRM1
SCHEMBL1663338 0.78 SIGMAR1 (0.59) CXCR4SIGMAR1MEN1CHRM2CHRM1
Hydrochloric Acid SCHEMBL28629993 0.77 CXCR4 (0.60) CXCR4SIGMAR1MEN1CHRM2CHRM1
Bromide SCHEMBL1257550 0.77 CXCR4 (0.78) CXCR4SIGMAR1MEN1CHRM2CHRM1
SCHEMBL5987431 0.76 DRD4 (0.64) ADH1BADH1CADH1AADH7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022178030-A1 TRPM8 AGONISTS AS COOLING AGENTS AND FOR THE TREATMENT OF DISEASE Concentric Analgesics, Inc. (US) 2022-08-25 WO disclosed