SCHEMBL24704369

SCHEMBL24704369

Bc1c[nH]c2nc(N)[nH]c(=O)c12

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.46
TYMS P04818 5/20 0.43
MAPT P10636 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GLA P06280 1/20 0.41
PMP22 Q01453 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18520454 0.80 DYRK1A (0.47) DYRK1ATYMSMAPTKDM4EALDH1A1
SCHEMBL15061831 0.79 TYMS (0.48) DYRK1ATYMSMAPTKDM4EALDH1A1
SCHEMBL12820951 0.79 DYRK1A (0.46) DYRK1ATYMS
SCHEMBL12884842 0.79 TYMS (0.46) DYRK1ATYMSMAPTKDM4EALDH1A1
SCHEMBL22227944 0.78 TYMS (0.50) DYRK1ATYMS
SCHEMBL13833421 0.78 TYMS (0.45) DYRK1ATYMS
SCHEMBL166747 0.76 TYMS (0.49) TYMS
SCHEMBL21161374 0.76 TYMS (0.49) TYMS
SCHEMBL25388812 0.76 TYMS (0.41) DYRK1ATYMS
SCHEMBL24233231 0.76 TYMS (0.41) DYRK1ATYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220396830-A1 BIOLUMINESCENT DETECTION OF DNA SYNTHESIS PROMEGA CORPORATION 2022-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220396830-A1 BIOLUMINESCENT DETECTION OF DNA SYNTHESIS RNGTT, NUDT1, DNTT DYRK1A 4489/4885TYMS 141/4885MAPT 4794/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.