SCHEMBL2472008

SCHEMBL2472008

Cc1nc2c([nH]1)c(=O)n(C)c(=O)n2CC=C=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 3/20 0.61
PDE1B Q01064 3/20 0.61
PDE1C Q14123 3/20 0.61
PDE2A O00408 2/20 0.61
MEN1 O00255 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2C19 P33261 2/20 0.52
BLM P54132 2/20 0.52
KMT2A Q03164 2/20 0.52
LMNA P02545 1/20 0.52
CYP1A1 P04798 1/20 0.52
NFKB1 P19838 1/20 0.52
MAPK1 P28482 1/20 0.52
PMP22 Q01453 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HIF1A Q16665 1/20 0.52
PDE5A O76074 2/20 0.42
TSHR P16473 1/20 0.41
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2948025 0.81 PDE1A (0.61) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL25249437 0.79 PDE1A (0.69) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL897036 0.76 PDE1A (1.00) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL461786 0.74 PDE2A (0.62) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL9122584 0.74 PDE1A (0.63) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL9803391 0.74 PDE1A (0.59) PDE1APDE1BPDE1CPDE2AMEN1
Verofylline SCHEMBL636856 0.73 PDE1A (0.78) PDE1APDE1BPDE1CPDE2AMEN1
Water SCHEMBL28799658 0.73 PDE2A (0.60) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL5688395 0.72 PDE2A (0.60) PDE1APDE1BPDE1CPDE2AMEN1
SCHEMBL9122677 0.71 ADORA2B (0.55) PDE1APDE1BPDE1CPDE2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011108001-A2 PROCESS FOR THE PREPARATION OF METHYL-METHYL-3, 4-DIHYDRO-2H-PYRAN-5-CARBOXYLATE SPC LIFESCIENCES PVT LTD (IN) 2011-09-09 WO disclosed
US-5498802-A 6-CHLORO-HEXANONE/2-/ FROM DEHYDRATION OF CYCLOHEXANOL TO CYCLOHEXENE AND REARRANGEMENTS, ALKALI METAL HYPOCHLORITE HOECHST CELANESE CORPORATION (US) 1996-03-12 US disclosed
US-5491265-A OXIDIZING WITH OZONE TO FORM 1-METHYLCYCLOPENTANOL, REACTING WITH ALKALI METAL HYPOCHLORITE, HEATING HOECHST CELANESE CORPORATION (US) 1996-02-13 US disclosed
US-4289776-A VASODILATORS, FIBRINOLYTIC HOECHST AKTIENGESELLSCHAFT (DE) 1981-09-15 US disclosed