SCHEMBL24743239

SCHEMBL24743239

COc1cccc(C(=O)N2CCC3(CCN(c4ccc(/C(C=N)=C/N)cc4)C3=O)C2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.44
PARP14 Q460N5 1/20 0.43
PARP10 Q53GL7 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
ALDH1A1 P00352 3/20 0.41
ABL1 P00519 4/20 0.41
BCR P11274 4/20 0.41
LMNA P02545 1/20 0.41
USP30 Q70CQ3 1/20 0.40
HSD11B1 P28845 1/20 0.39
MGLL Q99685 1/20 0.39
HPGD P15428 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24742760 0.95 L3MBTL1 (0.48) L3MBTL1PARP14PARP10CA12CA1
SCHEMBL24742765 0.87 DDB1 (0.47) ALDH1A1USP30TSHRITGB3ITGA2B
SCHEMBL24742759 0.81 ITGB3 (0.50) ITGB3ITGA2B
SCHEMBL24743004 0.81 ITGB3 (0.41) LMNAHPGDTSHRITGB3ITGA2B
SCHEMBL24743245 0.80 MAPT (0.46) L3MBTL1PARP14PARP10CA12CA1
SCHEMBL22355671 0.79 ITGB3 (0.37) ITGB3ITGA2B
SCHEMBL24742998 0.79 TSHR (0.45) CA12CA1CA2CA7CA9
SCHEMBL23529077 0.77 ROCK2 (0.57)
SCHEMBL24743008 0.77 ALDH1A1 (0.41) L3MBTL1ALDH1A1HPGDTP53TSHR
SCHEMBL24743010 0.75 ITGB3 (0.44) HPGDITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704121-B1 DIAZASPIRO ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-12-21 EP disclosed