Clopirac

Clopirac

SCHEMBL24768

Cc1cc(CC(=O)O)c(C)n1-c1ccc(Cl)cc1

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.61
ALDH1A1 P00352 1/20 0.58
MAPK1 P28482 2/20 0.55
NR1H4 Q96RI1 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
POLB P06746 1/20 0.50
USP14 P54578 1/20 0.49
USP7 Q93009 1/20 0.49
MAPT P10636 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KLKB1 P03952 1/20 0.47
CTSB P07858 1/20 0.47
SHMT2 P34897 1/20 0.47
PTGS2 P35354 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clopirac SCHEMBL28121041 0.90 NOTUM (0.51) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
SCHEMBL12608916 0.88 NOTUM (0.57) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
SCHEMBL11377279 0.87 NOTUM (0.56) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
Delmetacin SCHEMBL9446710 0.80 ABCB1 (0.73) MAPTNPSR1PTGS2
SCHEMBL16752445 0.80 NOTUM (0.49) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
SCHEMBL11257155 0.77 POLB (0.51) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
SCHEMBL1980763 0.76 NOTUM (1.00) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
SCHEMBL12608917 0.76 SHMT2 (0.46) NOTUMALDH1A1MAPK1SMN1; SMN2POLB
SCHEMBL19298013 0.74 NOTUM (0.48) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2
SCHEMBL13739403 0.74 ALDH1A1 (1.00) NOTUMALDH1A1MAPK1NR1H4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5908 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
US-RE50218-E1 Non-steroidal anti-inflammatory ophthalmic compositions SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2024-11-26 US claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
WO-2023142996-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT 上海岸阔医药科技有限公司 2023-08-03 WO claimed
EP-4034087-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS Research Inc. (CA) 2022-08-03 EP claimed
US-20220218611-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2022-07-14 US claimed
EP-3998932-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS Parsons, C. Lowell (US) 2022-05-25 EP claimed
US-20220110979-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC 2022-04-14 US claimed
US-5330981-A Antiinflammatory agents ISTITUTO GENTILI S.P.A. (IT) 1994-07-19 US claimed
EP-0569411-A1 ACYLAMINO-ALKYLIDEN-HYDROXY-BISPHOSPHONIC ACIDS USEFUL IN THE THERAPY OF OSTEOARTICULAR DISEASES. GENTILI IST SPA (IT) 1993-11-18 EP claimed
EP-0537313-A1 ARYLALKYL ESTERS OF 4,5-DIHYDROXY-9,10-DIHYDRO-9,10-DIOXO-2-ANTHRACENECARBOXYLIC ACID HAVING THERAPEUTICAL ACTIVITY. GENTILI IST SPA (IT) 1993-04-21 EP claimed
WO-1992019584-A1 ARYLALKYL ESTERS OF 4,5-DIHYDROXY-9,10-DIHYDRO-9,10-DIOXO-2-ANTHRACENECARBOXYLIC ACID HAVING THERAPEUTICAL ACTIVITY ISTITUTO GENTILI S.P.A. (IT) 1992-11-12 WO claimed
WO-1992013864-A1 ACYLAMINO-ALKYLIDEN-HYDROXY-BISPHOSPHONIC ACIDS USEFUL IN THE THERAPY OF OSTEOARTICULAR DISEASES ISTITUTO GENTILI S.P.A. (IT) 1992-08-20 WO claimed
EP-0452908-A2 Lipoxygenase-inhibiting compounds derived from non-steroidal antiinflammatory carboxylic acids ABBOTT LABORATORIES (US) 1991-10-23 EP claimed
US-5032588-A Non-steroidal antiinflammatory ABBOTT LABORATORIES (US) 1991-07-16 US claimed
WO-1991008744-A1 THIAZOLE LIPOXYGENASE-INHIBITING COMPOUNDS DERIVED FROM NON-STEROIDAL ANTIINFLAMMATORY CARBOXYLIC ACIDS ABBOTT LABORATORIES (US) 1991-06-27 WO claimed
EP-0408496-A2 Solid dosage form for pharmaceutical substances CIBA-GEIGY AG (CH) 1991-01-16 EP claimed
EP-0374602-A1 Lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1990-06-27 EP claimed