SCHEMBL2476855

SCHEMBL2476855

CCCCn1ccc2cccc(C#N)c21

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.38
CDK4 P11802 3/20 0.38
CCND1 P24385 3/20 0.38
CNR2 P34972 5/20 0.36
P2RX7 Q99572 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 1/20 0.35
APP P05067 1/20 0.34
GRK6 P43250 1/20 0.33
AR P10275 1/20 0.33
CTSL P07711 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27827799 0.78 P2RX7 (0.53) CDK4CCND1CNR2P2RX7KMT2A
SCHEMBL27844923 0.76 MAPT (0.44) CNR2MEN1LMNAHTTKMT2A
SCHEMBL17069069 0.75 XDH (0.39) MEN1LMNAHTTKMT2ASMN1; SMN2
SCHEMBL28990233 0.75 OXER1 (0.46) CDK4CCND1CNR2P2RX7
SCHEMBL15112345 0.74 CNR2 (0.56) CDK4CCND1CNR2DRD2DRD3
SCHEMBL17023237 0.73 LMNA (0.45) GRM2MEN1LMNAHTTKMT2A
SCHEMBL2872955 0.73 KMT2A (0.51) MEN1LMNAHTTKMT2ATSHR
SCHEMBL3821765 0.72 GRM2 (0.44) GRM2CNR2MEN1LMNAHTT
SCHEMBL9684661 0.71 GRK6 (0.39) GRM2DRD2DRD3MEN1LMNA
SCHEMBL22871225 0.70 HTR2A (0.42) DRD2DRD3MEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362874-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2011-09-07 EP disclosed